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GSK3 Degrader PT-65

 

CAS: 2721998-87-2

 

Chemical Name: 3-Amino-6-(4-((4-(4-(1-(17-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)-3,6,9,12,15-pentaoxaheptadecyl)-1H-1,2,3-triazol-4-yl)butyl)piperazin-1-yl)sulfonyl)phenyl)-N-(pyridin-3-yl)pyrazine-2-carboxamide

 

 
GLXC-26356For Lab R&D Uses Only
        Cat No: GLXC-26356

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent GSK3 Degrader (DC50 = 28.3 nM and 34.2 nM against GSK3α and GSK3β, respectively)

 

Ref: https://www.sciencedirect.com/science/article/abs/pii/S0223523421007388


Analytical data click for PDF file

 

 

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