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 PT2399

 

CAS: 1672662-14-4

 

Chemical Name: 3-[(1S)-7-(Difluoromethylsulfonyl)-2,2-difluoro-1-hydroxy-indan-4-yl]oxy-5-fluoro-benzonitrile

 

 

GLXC-09305        Cat No: GLXC-09305

                 For Lab R&D Uses Only

 

Purity:               > 98% (HPLC)

Storage:             Refrigerator (4 °C)

 


Product Description:

Novel HIF2alpha antagonist, causing tumor regression in preclinical models of primary and metastatic pVHL-defective ccRCC in an on-target fashion

 

References:

1) https://www.pnas.org/content/115/52/13240.long

2) https://onlinelibrary.wiley.com/doi/abs/10.1002/jmr.2730

3) https://cancerres.aacrjournals.org/content/77/22/6321.long

 

Analytical data click for PDF file

 

 

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