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CAS: N/A
Chemical Name: 6-(4-Chloro-2-methylphenyl)-5-(5-chloro-2-methylphenyl)-2-(2,4-dimethoxypyrimidin-5-yl)-1-isopropyl-5,6-dihydropyrrolo[3,4-d]imidazol-4(1H)-one
Purity: >98% (HPLC)
Novel, highly potent p53-MDM2 inhibitor with an IC50 value of 0.08 nmol/L, displaying excellent oral efficacy in the human SJSA1-based xenograft model.
Ref: https://pubs.acs.org/doi/abs/10.1021/acs.jmedchem.7b00104
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