Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2326521-71-3
Chemical Name: Adagrasib; MRTX-849; 2-[(2S)-4-[7-(8-Chloronaphthalen-1-yl)-2-[[(2S)-1-methylpyrrolidin-2-yl]methoxy]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]-1-(2-fluoroprop-2-enoyl)piperazin-2-yl]acetonitrile
Purity: >98% (HPLC)
Novel covalent inhibitor of KRASG12C
References:
1) https://pubs.acs.org/doi/10.1021/acs.jmedchem.9b02052
2) https://onlinelibrary.wiley.com/doi/full/10.1111/joim.13057
3) https://cancerdiscovery.aacrjournals.org/content/10/1/54.long
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