Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 761436-62-8
Chemical Name: TAC544; 2-[[5-Bromo-2-[[2-methoxy-4-(4-morpholinyl)phenyl]amino]-4-pyrimidinyl]amino]-N-methyl-benzenesulfonamide
Purity: >98% (HPLC)
Novel focal adhesion kinase (FAK) inhibitor, potently blocking kinase activity of FAK along with Aurora A, activated Cdc42-associated kinase 1 (ACK1), Met, insulin receptor (IR), TrkA, and IGF-1R
References:
1) https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4365862/
2) https://www.ncbi.nlm.nih.gov/pmc/articles/PMC2287283/
3) https://www.mdpi.com/2072-6694/11/11/1683/pdf
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