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Glixx Laboratorie
CAS: 2316837-08-6
Chemical Name: (2S,4R)-N-((S)-3-(4-((4-(((1r,3r)-3-(3-Chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl)carbamoyl)phenyl)ethynyl)-[1,4'-bipiperidin]-1'-yl)-1-(4-(4-methylthiazol-5-yl)phenyl)-3-oxopropyl)-4-hydroxy-1-((R)-3-methyl-2-(3-methylisoxazol-5-yl)butanoyl)pyrrolidine-2-carboxamide
Purity: >98% (HPLC)
Novel highly potent PROTAC androgen receptor (AR) degrader, effectively inhibiting AR-positive breast cancer cell growth in vitro and tumor growth in vivo
References:
1) https://www.sciencedirect.com/science/article/pii/S1476558620301330
2) https://www.sciencedirect.com/science/article/pii/S1476558619304865
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