Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2574389-19-6
Chemical Name: (3S,6S,14S)-6-Acetamido-N-((S)-1-(benzo[d]thiazol-2-yl)-5-guanidino-1-oxopentan-2-yl)-3-isobutyl-9-methyl-2,5,8-trioxo-1,4,9-triazacyclotetradecane-14-carboxamide
Purity: >98% (HPLC)
Novel macrocyclic inhibitor of HGF-activating serine proteases, potently inhibiting matriptase and hepsin, overcoming resistance to receptor tyrosine kinase inhibitors and blocking lung cancer progression
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c01671
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