Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2866408-21-9
Chemical Name: N-(4-((1-Isopropylpiperidin-4-yl)amino)-6-methoxy-7-(3-(pyrrolidin-1-yl)propoxy)quinolin-2-yl)acrylamide
Purity: >98% (HPLC)
The first-in-class G9a/GLP covalent irreversible inhibitor, targeting a cysteine residue at the substrate binding site
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.2c00652
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