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CAS: N/A
Chemical Name: N-(2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)-2-((6-(4-(2-fluoro-5-((4-oxo-3,4-dihydrophthalazin-1-yl)methyl)benzoyl)piperazin-1-yl)-6-oxohexyl)amino)acetamide
Purity: >98% (HPLC)
Novel PARP1 degrader, inducing PARP1 protein degradation with DC50 values of 53 nM in MDA-MB-231 cells, exhibiting broad antiproliferative activities and bearing nearly 60-fold tumor-selectivity
Ref: https://www.sciencedirect.com/science/article/pii/S0968089622003017
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