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CAS: N/A
Chemical Name: N,N'-((2,2'-((Oxybis(ethane-2,1-diyl))bis(oxy))bis(acetyl))bis(piperidine-1,4-diyl))bis(4-((4-((4-chloro-3-((1,1-dimethylethyl)sulfonamido)phenyl)amino)-5-methylpyrimidin-2-yl)amino)-2-fluorobenzamide)
Purity: >98% (HPLC)
Novel Bivalent BET Bromodomain Inhibitor, Increasing Potency and Selectivity for BRDT via Protein Conformational Plasticity
Ref: https://pubs.acs.org/doi/abs/10.1021/acs.jmedchem.2c00453
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