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CAS: N/A
Chemical Name: 4-((4-((4-Chloro-3-((1,1-dimethylethyl)sulfonamido)phenyl)amino)-5-methylpyrimidin-2-yl)amino)-N-(1-(1-(3-((1,1-dimethylethyl)sulfonamido)-5-((2-((3-fluoro-4-(piperidin-4-ylcarbamoyl)phenyl)amino)-5-methylpyrimidin-4-yl)amino)phenyl)-1-oxo-5,8,11-trioxa-2-azatetradecan-14-oyl)piperidin-4-yl)-2-fluorobenzamide hydrochloride
Purity: >98% (HPLC)
Novel Bivalent BET Bromodomain Inhibitor, Increasing Potency and Selectivity for BRDT via Protein Conformational Plasticity
Ref: https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5457702/
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