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CAS: 2755823-12-0
Chemical Name: 3-Allyl-2-(((3R,5R)-5-(4-(benzyloxy)phenyl)-1-methylpiperidin-3-yl)amino)-3,5-dihydro-4H-pyrrolo[3,2-d]pyrimidin-4-one
Purity: >98% (HPLC)
Novel potent, selective and endogenous binder competitive inhibitor of SETDB1 tandem tudor domain (SETDB1-TTD) with a KD of 88 nM
Ref: https://onlinelibrary.wiley.com/doi/10.1002/anie.202017200
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