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AZ'3137

 

CAS: 2960179-55-7

 

Chemical Name: 4-(4-(4-(4-((4-(2-(2,6-Dioxopiperidin-3-yl)-7-methoxy-1-oxoisoindolin-5-yl)piperazin-1-yl)methyl)piperidin-1-yl)phenyl)piperidin-1-yl)-3-fluoro-2-(trifluoromethyl)benzonitrile

 

 
GLXC-28759For Lab R&D Uses Only
        Cat No: GLXC-28759

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel orally bioavailable androgen receptor (AR) degrader, showing degradation of AR and L702H mutant AR with good oral bioavailability across species

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c00269

 

Analytical data click for PDF file

 

 

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