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CAS: 2960179-55-7
Chemical Name: 4-(4-(4-(4-((4-(2-(2,6-Dioxopiperidin-3-yl)-7-methoxy-1-oxoisoindolin-5-yl)piperazin-1-yl)methyl)piperidin-1-yl)phenyl)piperidin-1-yl)-3-fluoro-2-(trifluoromethyl)benzonitrile
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel orally bioavailable androgen receptor (AR) degrader, showing degradation of AR and L702H mutant AR with good oral bioavailability across species
Reference:
https://pubs.acs.org/doi/10.1021/acs.jmedchem.4c00269
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