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JNJ-54082730

 

CAS: 2097493-39-3

 

Chemical Name: ((3S,4R)-3-(5-(Difluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl)-4-methylpiperidin-1-yl)(2,6-dimethylpyridin-4-yl)methanone

 

 
GLXC-28901For Lab R&D Uses Only
        Cat No: GLXC-28901

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel highly potent inhibitor of PDE2A with hPDE2A: IC50 = 0.9 (0.8 -1) nM, n= 93 [Mean (95% Confidence Interval)], Ki = 0.7 nM

 

Reference:

https://www.eubopen.org/sites/www.eubopen.org/files/chemical-probes/EUbOPEN_ProbeSheet_JNJ-54082730_v1.pdf

 

Analytical data click for PDF file

 

 

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