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CAS: 2766231-05-2 (free base: 2409538-60-7)
Chemical Name: XNW5004 maleate; N-((4,6-Dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-2-methyl-5-((1r,3r)-3-(piperidin-1-yl)cyclobutoxy)benzamide maleate
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel, selective, substrate-competitive inhibitor of EZH2, significantly suppressing level of H3K27Me3, arresting cell cycle in G1/S phase and promoting apoptosis in tumor
References:
https://ascopubs.org/doi/10.1200/JCO.2025.43.16_suppl.7012
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