Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 1429028-96-5
Chemical Name: 4,9-Bis((3-(4-methylpiperazin-1-yl)propyl)amino)-2,7-bis(3-morpholinopropyl)benzo[lmn][3,8]phenanthroline-1,3,6,8(2H,7H)-tetraone
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel BCL-2 quadruplex ligand, binding to quadruplex-forming promoter regions in a number of genes and down-regulating their transcription, showing significant in vivo anti-tumour activity against the MIA PaCa-2 pancreatic cancer xenograft model
References:
https://www.mdpi.com/1424-8247/15/1/7
https://www.nature.com/articles/srep11385
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