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Cloperastine hydrochloride

 

CAS: 14984-68-0

 

Chemical Name: 1-[2-[(4-Chlorophenyl)-phenylmethoxy]ethyl]piperidine Hydrochloride

 

 
GLXC-22767For Lab R&D Uses Only
        Cat No: GLXC-22767

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Antitussive and antihistamine agent as a σ1 receptor agonist (Ki = 20 nM), a GIRK channel blocker, a H1 receptor antagonist (Ki = 3.8 nM)

 

References:

1) https://www.nature.com/articles/s41419-020-02842-x

2) https://www.sciencedirect.com/science/article/abs/pii/S0028390820302823?via%3Dihub

3) https://www.sciencedirect.com/science/article/pii/S009130571630017X?via%3Dihub

 

Analytical data click for PDF file

 

 

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