Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2225938-86-1
Chemical Name: N-[(4,6-Dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[2-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]propanoylamino]ethyl]piperazin-1-yl]pyridin-3-yl]-1-propan-2-ylindazole-4-carboxamide
Purity: >98% (HPLC)
Novel fast-acting EZH2 degrader, effectively depleting both canonical EZH2-PRC2 and noncanonical EZH2-cMyc complexes, inducing leukaemia cell growth inhibition, apoptosis and cell cycle progression arrest
References:
https://pubmed.ncbi.nlm.nih.gov/?term=MS177&sort=date
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