Glixx Laboratories Inc

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ERB-2

 

CAS: N/A

 

Chemical Name: (2S,4R)-1-((S)-2-(tert-Butyl)-14-(2-hydroxy-5-(5-hydroxy-7-vinylbenzo[d]oxazol-2-yl)phenoxy)-4-oxo-6,9,12-trioxa-3-azatetradecanoyl)-4-hydroxy-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide

 

 
GLXC-90026For Lab R&D Uses Only
        Cat No: GLXC-90026

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel ERβ-targeting PROTAC, degrading ERβ in dose, time, and UPS dependent manner, inducing ROS accumulation in NSCLC cells and reversing Osimertinib resistance in vivo

 

Reference:

https://www.sciencedirect.com/science/article/abs/pii/S0045206825012544


Analytical data click for PDF file

 

 

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