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CAS: 2489876-41-5
Chemical Name: N-(4-(chlorodifluoromethoxy)phenyl)-6-((2-(2-(((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-2-oxoethoxy)ethyl)amino)-5-(1H-pyrazol-5-yl)nicotinamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel potent BCR-Abl PROTAC, inducing degradation and demonstrating in vivo activity
Ref: https://pubs.rsc.org/en/content/articlelanding/2020/cc/d0cc02201b#!divAbstract
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