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CAS: N/A
Chemical Name: 2-((7-Acetyl-3-(furan-2-ylmethyl)-4-oxo-3,4,5,6,7,8-hexahydropyrido[4',3':4,5]thieno[2,3-d]pyrimidin-2-yl)thio)-N-(2-methylpyridin-3-yl)acetamide
Purity: >98% (HPLC)
Novel potent inhibitor of BET proteins with a preferential and 475-fold selectivity for the second bromodomain of the BRD3 protein (BRD3-BDII) over its first bromodomain (BRD3-BDI)
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c02168
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