Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2417917-17-8
Chemical Name: 1-[(3S)-4-[7-[6-Amino-4-methyl-3-(trifluoromethyl)pyridin-2-yl]-6-chloro-8-fluoro-2-[[(2S)-1-methylpyrrolidin-2-yl]methoxy]quinazolin-4-yl]-3-methylpiperazin-1-yl]prop-2-en-1-one
Purity: >98% (HPLC)
Novel covalent allosteric KRASG12C inhibitor
References:
1) https://www.nature.com/articles/s41417-021-00383-9
2) https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.1c00389
3) https://ascopost.com/issues/september-10-2020/targeting-kras-mutated-tumors/
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