Glixx Laboratories Inc

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Enbezotinib

 

CAS: 2359649-81-1 (2411115-73-4)

 

Chemical Name: TPX-0046; (13E,14E,15aR,18aS,5S)-35-Fluoro-5-methyl-15,15a,16,17,18,18a-hexahydro-4-oxa-7-aza-1(5,3)-cyclopenta[b]pyrazolo[1',5':1,2]pyrimido[4,5-e][1,4]oxazina-3(3,2)-pyridinacyclooctaphan-8-one

 

 
GLXC-25750For Lab R&D Uses Only
        Cat No: GLXC-25750

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent RET/SRC inhibitor with a mean IC50 of 17 nM for RETG810R in Ba/F3 cell proliferation assay

 

Ref: https://link.springer.com/article/10.1007/s10637-022-01259-x

 

Analytical data click for PDF file

 

 

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