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Glixx Laboratorie
CAS: N/A
Chemical Name: (Z)-2-(2,6-Dioxopiperidin-3-yl)-N-(8-(5-(4-isopropylbenzylidene)-2,4-dioxothiazolidin-3-yl)octyl)-1,3-dioxoisoindoline-5-carboxamide
Purity: >98% (HPLC)
Novel MYC PROTAC, inducing Cereblon-dependent degradation of MYC, GSPT1/2, and PLK1, showing cellular activity in conventional gastrointestinal cancer cell lines and primary cancer organoids
Ref: https://www.sciencedirect.com/science/article/pii/S004520682100883X
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