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CAS: 2756388-01-7
Chemical Name: N-(5-((5-(4-Acetylpiperazine-1-carbonyl)-4-methoxy-2-methylphenyl)thio)thiazol-2-yl)-4-(4-(7-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamido)heptyl)piperazin-1-yl)benzamide
Purity: >98% (HPLC)
Novel ITK-selective degrader, suppressing canonical NF-κB pathway and GATA-3 expression, overcoming chemotherapy resistance in T cell lymphomas
Reference:
https://www.cell.com/cell-chemical-biology/fulltext/S2451-9456(23)00086-7
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