Glixx Laboratories Inc
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Glixx Laboratorie
CAS: 2406278-81-5
Chemical Name: N-((1R,3r)-3-(5-(5-Ethoxypyridin-2-yl)-4-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl)cyclobutyl)quinoxaline-5-carboxamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel highly potent tankyrase inhibitor, showing picomolar IC50 inhibition in a cellular (HEK293) WNT/β-catenin signaling reporter assay, no off-target liabilities, overall favorable absorption, distribution, metabolism, and excretion (ADME) properties, and an improved pharmacokinetic profile in mice
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c01264
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