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CAS: N/A
Chemical Name: Cyclo[(R)-2-(4-(2-imino-3-amino-3-oxopropyl)-1H-1,2,3-triazol-1-yl)acetyl-Val-Trp-Phe-Gly-homoVal-(m-CF3)Phe-(1-Bz-4-NH)Pro]
Purity: >98% (HPLC)
Neutral MDM2-p53 Inhibitor, inhibiting MDM2-p53 interaction with an IC50 of 8.9 nM
Reference:
https://pubs.acs.org/doi/abs/10.1021/acsmedchemlett.3c00117
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