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CAS: N/A
Chemical Name: 6-((5-Cyclopropyl-1H-pyrazol-3-yl)amino)-2-(4-(3-formyl-4-hydroxybenzyl)piperazin-1-yl)-N-(prop-2-yn-1-yl)pyrimidine-4-carboxamide
Purity: >98% (HPLC)
Novel reversible lysine-targeted probe, revealing residence time-based kinase selectivity, targeting Aurora A and showing sustained, quasi-irreversible occupancy in vivo
Ref: https://www.nature.com/articles/s41589-022-01019-1
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