Glixx Laboratories Inc

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Glixx Laboratorie

 

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Etavopivat

 

CAS: 2245053-57-8

 

Chemical Name: FT-4202; (2S)-1-[5-(2,3-Dihydro-[1,4]dioxino[2,3-b]pyridin-7-ylsulfonyl)-1,3,4,6-tetrahydropyrrolo[3,4-c]pyrrol-2-yl]-3-hydroxy-2-phenylpropan-1-one

 

 
GLXC-25164For Lab R&D Uses Only
        Cat No: GLXC-25164

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel oral pyruvate kinase (PKR) activator, showing potent antisickling effects and improving RBC survival and Hb levels in SCA mice

 

References:

1) https://accp1.onlinelibrary.wiley.com/doi/10.1002/cpdd.1058

2) https://jpet.aspetjournals.org/content/early/2022/01/14/jpet.121.000743

3) https://ashpublications.org/bloodadvances/article/5/9/2385/475849/

 

Analytical data click for PDF file

 

 

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