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CAS: N/A
Chemical Name: N-(1-(2-Ethynylthiazole-4-carbonyl)-4-(1-methyl-1H-benzo[d]imidazol-2-yl)piperidin-4-yl)-2-phenylthiazole-5-carboxamide
For Lab R&D Uses Only
Purity: >98% (HPLC)
Novel reversible covalent STING antagonist, maintaining activity against the most prevalent human STING variant (R232), effectively suppressing STING signaling in primary human CD14+ monocytes, and exhibiting moderate metabolic stability
Reference:
https://pubs.acs.org/doi/10.1021/acsmedchemlett.5c00611
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