Glixx Laboratories Inc

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PROTAC HL-8

 

CAS: 2766352-64-9

 

Chemical Name: PI3K degrader HL-8; (2R,4S)-1-((S)-2-(7-(2-(5-(6-(5-((2,4-Difluorophenyl)sulfonamido)-6-methoxypyridin-3-yl)imidazo[1,2-a]pyridin-3-yl)-1,3,4-oxadiazol-2-yl)benzamido)heptanamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide

 

 
GLXC-25659For Lab R&D Uses Only
        Cat No: GLXC-25659

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel PI3K degrader, showing a significant and complete degradation effect on PI3K kinase at a concentration of 10 μM within 8 h

 

Ref: https://www.sciencedirect.com/science/article/abs/pii/S0968089622000992

 

Analytical data click for PDF file

 

 

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