Glixx Laboratories Inc

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Glixx Laboratorie

 

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Sunvozertinib

 

CAS: 2370013-12-8

 

Chemical Name: DZD9008; N-[5-[[4-[5-Chloro-4-fluoro-2-(2-hydroxypropan-2-yl)anilino]pyrimidin-2-yl]amino]-2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-4-methoxyphenyl]prop-2-enamide

 

 
GLXC-25829For Lab R&D Uses Only
        Cat No: GLXC-25829

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel potent ErbBs (EGFR, Her2, especially mutant forms) inhibitor, showing IC50s of 20.4, 20.4, 1.1, 7.5, and 80.4 nM for EGFR exon 20 NPH insertion, EGFR exon 20 ASV insertion, EGFR L858R and T790M mutations, and Her2 Exon20 YVMA, and EGFR WT A431, respectively, also inhibiting BTK

 

References:

1) https://www.tandfonline.com/doi/abs/10.1080/03007995.2022.2083326

2) https://aacrjournals.org/cancerdiscovery/article/doi/10.1158/2159-8290.CD-21-1615/694369/Sunvozertinib-a-selective-EGFR-inhibitor-for

 

Analytical data click for PDF file

 

 

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