Glixx Laboratories Inc

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Glixx Laboratorie

 

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GNE-7883

 

CAS: 2648450-42-2

 

Chemical Name: 5-(4-Cyclohexylphenyl)-3-(3-(fluoromethyl)azetidine-1-carbonyl)-2-(3-methylpyrazin-2-yl)pyrazolo[1,5-a]pyrimidin-7(4H)-one

 

 
GLXC-27634For Lab R&D Uses Only
        Cat No: GLXC-27634

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

Novel allosteric pan-TEAD inhibitor, blocking oncogenic YAP/TAZ signaling and overcoming KRAS G12C inhibitor resistance

 

Reference:

https://www.nature.com/articles/s43018-023-00577-0


 

Analytical data click for PDF file

 

 

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