Glixx Laboratories Inc

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YM458

 

CAS: 2770108-93-3

 

Chemical Name: (S)-4'-((5-(2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetamido)pentyl)oxy)-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-5-(ethyl(tetrahydro-2H-pyran-4-yl)amino)-4-methyl-[1,1'-biphenyl]-3-carboxamide

 

 
GLXC-25680For Lab R&D Uses Only
        Cat No: GLXC-25680

 

Purity:               >98% (HPLC)

Storage:             Refrigerator (4 °C)

 

 

Product Description:

First-in-class dual EZH2/BRD4 inhibitor, displaying potent inhibitory activity against EZH2 and BRD4 and remarkable antiproliferative capacity against 11 solid cancer cell lines

 

Reference:

https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c01876

 

Analytical data click for PDF file

 

 

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