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CAS: 2426628-52-4
Chemical Name: 10,13-Dimethyl-9-oxo-3-(trifluoromethyl)-4,5,10,12,13,18,20-heptazapentacyclo[14.5.2.12,5.011,15.019,22]tetracosa-1(21),2(24),3,11,14,16(23),17,19(22)-octaene-14-carbonitrile
Purity: >98% (HPLC)
Novel selective inhibitor of DYRK1A/B, demonstrating antitumor efficacy in head and neck squamous cell carcinoma (HNSCC) cell lines
Reference:
https://pubs.acs.org/doi/10.1021/acsmedchemlett.1c00630
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