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Glixx Laboratorie
CAS: N/A
Chemical Name: (Z)-3-((1H-Indol-2-yl)methylene)-4-((4-hydroxypiperidin-4-yl)ethynyl)indolin-2-one
Purity: >98% (HPLC)
Novel potent and selective serine-threonine kinase TAO3 inhibitor (IC50= 42 nM against TAO3, IC50=237 nM against MEKK3)
Ref: https://aacrjournals.org/cancerres/article/81/6/1472/670547
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