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CAS: 2369022-68-2
Chemical Name: 2-(4-(1-(1-(4-((4R,5S)-4,5-bBs(4-chlorophenyl)-2-(2-isopropoxy-4-methoxyphenyl)-4,5-dihydro-1H-imidazole-1-carbonyl)-2-oxopiperazin-1-yl)-2-oxo-6,9,12,15-tetraoxa-3-azaheptadecan-17-yl)-1H-1,2,3-triazol-4-yl)phenyl)-2H-indazole-7-carboxamide
Purity: >98% (HPLC)
Novel poly (ADP-ribose) polymerase-1 (PARP1) degrader, inducing significant PARP1 cleavage and programmed cell death in the MDA-MB-231 cell line
Ref: https://pubs.rsc.org/en/content/articlelanding/2019/CC/C8CC07813K
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