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CAS: 2484739-25-3
Chemical Name: 3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-[1-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperidin-4-yl]-N-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamide
Purity: >98% (HPLC)
Novel potent and selective heterobifunctional degrader of p300/CBP
References:
1) https://www.cell.com/cell-chemical-biology/fulltext/S2451-9456(21)00154-9
2) https://www.cell.com/cell-chemical-biology/fulltext/S2451-9456(20)30513-4
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