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CAS: N/A
Chemical Name: JMV-3168; (R)-N-(2-(1H-Indol-3-yl)-1-(4-(4-methoxybenzyl)-5-phenethyl-4H-1,2,4-triazol-3-yl)ethyl)tetrahydro-2H-pyran-4-carboxamide
Purity: >98% (HPLC)
Novel ghrelin receptor (GHS-R1a) antagonist [IC50 (affinity): 5 nM IC50 (Ca2+ ): 60 nM]
Ref: https://pubs.acs.org/doi/10.1021/acs.jmedchem.1c02191
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